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Assay Detail

CHEMBL872359

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition constant against Dopamine receptor D2 in olfactory bulbectomized rat
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Rattus norvegicus
Confidence 9 — Direct single protein target
Curated By Expert

Target

D(2) dopamine receptor (CHEMBL339)
Type SINGLE PROTEIN
Organism Rattus norvegicus

Publication

Designed multiple ligands. An emerging drug discovery paradigm.
Morphy R, Rankovic Z.
J Med Chem (2005) 48 : 6523 -6543
PubMed 16220969 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 7.28 7.28

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL268258 1 7.28

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL268258 Ki = 52.0 nM 7.28