Assay Detail
Functional
CHEMBL877774
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antinociceptive activity determined in vivo in tail flick assay in male Swiss mice with saline
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Mus musculus |
| Tissue | Tail |
| Confidence | 1 — Organism |
| Curated By | Intermediate |
Publication
Non-peptide ligands for opioid receptors. Design of kappa-specific agonists.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 9.00 | 9.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL70 | MORPHINE | 4.0 | 1 | 9.00 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL70 | MORPHINE | Ki | = | 1.0 | nM | 9.00 |