Assay Detail
Binding
CHEMBL881485
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Inhibitory activity against Mitogen-activated protein kinase 14, p38-alpha
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Expert |
Publication
Fast small molecule similarity searching with multiple alignment profiles of molecules represented in one-dimension.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 6.45 | 7.05 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL423781 | — | — | 1 | 7.05 |
| CHEMBL328126 | — | — | 1 | 5.85 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL423781 | — | IC50 | = | 90.0 | nM | 7.05 |
| CHEMBL328126 | — | IC50 | = | 1400.0 | nM | 5.85 |