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Assay Detail

CHEMBL882391

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of [3H]citalopram binding to the serotonin transporter in rhesus (Macaca mulatta) or cynomolgus monkey (Macaca fascicularis) caudate-putamen.
50
Total Activities
35
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Cercopithecidae
Tissue Caudate-putamen
Confidence 8 — Homologous single protein target
Curated By Expert

Target

Sodium-dependent serotonin transporter (CHEMBL228)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Synthesis of 6- and 7- hydroxy-8-azabicyclo[3.2.1]octanes and their binding affinity for the dopamine and serotonin transporters.
Meltzer PC, Wang B, Chen Z, Blundell P, Jayaraman M, Gonzalez MD, George C, Madras BK.
J Med Chem (2001) 44 : 2619 -2635
PubMed 11472216 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 50 6.32 8.66

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL87567 2 8.66
CHEMBL87031 2 8.61
CHEMBL86654 2 8.25
CHEMBL91184 1 7.82
CHEMBL330228 3 7.56
CHEMBL315172 2 7.47
CHEMBL86590 2 7.01
CHEMBL84680 1 6.96
CHEMBL2310846 2 6.86
CHEMBL2079586 2 6.80
CHEMBL421167 2 6.78
CHEMBL316428 1 6.58
CHEMBL2114227 1 6.54
CHEMBL421546 1 6.17
CHEMBL88915 1 6.06
CHEMBL89476 1 6.00
CHEMBL606929 1 5.91
CHEMBL606928 1 5.80
CHEMBL432571 1 5.48
CHEMBL89906 1 5.31
CHEMBL606930 1 5.27
CHEMBL314887 2 5.24
CHEMBL2115225 1 5.15
CHEMBL89469 1 5.10
CHEMBL314912 1 5.02
CHEMBL88246 1 4.97
CHEMBL89662 1 4.54
CHEMBL89208 3 4.06
CHEMBL89709 2 -
CHEMBL330250 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL87567 IC50 = 2.19 nM 8.66
CHEMBL87031 IC50 = 2.47 nM 8.61
CHEMBL86654 IC50 = 5.57 nM 8.25
CHEMBL87567 IC50 = 5.95 nM 8.22
CHEMBL91184 IC50 = 15.0 nM 7.82
CHEMBL330228 IC50 = 27.7 nM 7.56
CHEMBL87031 IC50 = 27.7 nM 7.56
CHEMBL315172 IC50 = 34.2 nM 7.47
CHEMBL86654 IC50 = 94.0 nM 7.03
CHEMBL86590 IC50 = 97.0 nM 7.01
CHEMBL84680 IC50 = 109.0 nM 6.96
CHEMBL2310846 IC50 = 139.0 nM 6.86
CHEMBL2079586 IC50 = 160.0 nM 6.80
CHEMBL421167 IC50 = 166.0 nM 6.78
CHEMBL315172 IC50 = 180.0 nM 6.75
CHEMBL316428 IC50 = 260.0 nM 6.58
CHEMBL2114227 IC50 = 290.0 nM 6.54
CHEMBL330228 IC50 = 533.0 nM 6.27
CHEMBL421546 IC50 = 677.0 nM 6.17
CHEMBL88915 IC50 = 867.0 nM 6.06
CHEMBL89476 IC50 = 991.0 nM 6.00
CHEMBL2079586 IC50 = 1130.0 nM 5.95
CHEMBL606929 IC50 = 1220.0 nM 5.91
CHEMBL330228 IC50 = 1390.0 nM 5.86
CHEMBL421167 IC50 = 1450.0 nM 5.84
CHEMBL606928 IC50 = 1590.0 nM 5.80
CHEMBL86590 IC50 = 2520.0 nM 5.60
CHEMBL432571 IC50 = 3320.0 nM 5.48
CHEMBL89906 IC50 = 4850.0 nM 5.31
CHEMBL2310846 IC50 = 5300.0 nM 5.28
CHEMBL606930 IC50 = 5370.0 nM 5.27
CHEMBL314887 IC50 = 5820.0 nM 5.24
CHEMBL2115225 IC50 = 7038.0 nM 5.15
CHEMBL89469 IC50 = 7990.0 nM 5.10
CHEMBL314912 IC50 = 9560.0 nM 5.02
CHEMBL88246 IC50 = 10700.0 nM 4.97
CHEMBL89662 IC50 = 28600.0 nM 4.54
CHEMBL89208 IC50 = 88000.0 nM 4.06
CHEMBL89709 IC50 > 10000.0 nM -
CHEMBL314887 IC50 > 20000.0 nM -
CHEMBL88563 IC50 > 10000.0 nM -
CHEMBL89208 IC50 > 20000.0 nM -
CHEMBL314138 IC50 > 10000.0 nM -
CHEMBL88563 IC50 > 100000.0 nM -
CHEMBL89754 IC50 > 10000.0 nM -
CHEMBL86710 IC50 > 6000.0 nM -
CHEMBL89756 IC50 > 100000.0 nM -
CHEMBL89208 IC50 > 10000.0 nM -
CHEMBL330250 IC50 > 20000.0 nM -
CHEMBL89709 IC50 > 20000.0 nM -