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Assay Detail

CHEMBL890059

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Binding
Binding affinity to rat SERT
30
Total Activities
30
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Rattus norvegicus
Confidence 9 — Direct single protein target
Curated By Expert

Target

Sodium-dependent serotonin transporter (CHEMBL313)
Type SINGLE PROTEIN
Organism Rattus norvegicus

Publication

Dual serotonin transporter/histamine H3 ligands: Optimization of the H3 pharmacophore.
Keith JM, Gomez LA, Letavic MA, Ly KS, Jablonowski JA, Seierstad M, Barbier AJ, Wilson SJ, Boggs JD, Fraser IC, Mazur C, Lovenberg TW, Carruthers NI.
Bioorg Med Chem Lett (2007) 17 : 702 -706
PubMed 17107798 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 30 8.36 9.14

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL396945 1 9.14
CHEMBL234526 1 9.00
CHEMBL394787 1 8.89
CHEMBL394800 1 8.85
CHEMBL396459 1 8.82
CHEMBL233054 1 8.80
CHEMBL394861 1 8.70
CHEMBL233471 1 8.70
CHEMBL396703 1 8.70
CHEMBL427845 1 8.66
CHEMBL396981 1 8.57
CHEMBL41 FLUOXETINE 4.0 1 8.55
CHEMBL232660 1 8.52
CHEMBL395022 1 8.48
CHEMBL233053 1 8.32
CHEMBL242820 1 8.28
CHEMBL394801 1 8.28
CHEMBL242817 1 8.24
CHEMBL395096 1 8.24
CHEMBL234525 1 8.20
CHEMBL232661 1 8.12
CHEMBL234732 1 8.10
CHEMBL232218 1 8.08
CHEMBL245130 1 8.00
CHEMBL233470 1 8.00
CHEMBL232620 1 7.82
CHEMBL232621 1 7.82
CHEMBL233681 1 7.72
CHEMBL429440 1 7.68
CHEMBL232010 1 7.60

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL396945 Ki = 0.73 nM 9.14
CHEMBL234526 Ki = 1.0 nM 9.00
CHEMBL394787 Ki = 1.3 nM 8.89
CHEMBL394800 Ki = 1.4 nM 8.85
CHEMBL396459 Ki = 1.5 nM 8.82
CHEMBL233054 Ki = 1.6 nM 8.80
CHEMBL394861 Ki = 2.0 nM 8.70
CHEMBL233471 Ki = 2.0 nM 8.70
CHEMBL396703 Ki = 2.0 nM 8.70
CHEMBL427845 Ki = 2.2 nM 8.66
CHEMBL396981 Ki = 2.7 nM 8.57
CHEMBL41 FLUOXETINE Ki = 2.8 nM 8.55
CHEMBL232660 Ki = 3.0 nM 8.52
CHEMBL395022 Ki = 3.3 nM 8.48
CHEMBL233053 Ki = 4.8 nM 8.32
CHEMBL242820 Ki = 5.3 nM 8.28
CHEMBL394801 Ki = 5.3 nM 8.28
CHEMBL242817 Ki = 5.7 nM 8.24
CHEMBL395096 Ki = 5.7 nM 8.24
CHEMBL234525 Ki = 6.3 nM 8.20
CHEMBL232661 Ki = 7.6 nM 8.12
CHEMBL234732 Ki = 8.0 nM 8.10
CHEMBL232218 Ki = 8.4 nM 8.08
CHEMBL245130 Ki = 10.0 nM 8.00
CHEMBL233470 Ki = 10.0 nM 8.00
CHEMBL232620 Ki = 15.0 nM 7.82
CHEMBL232621 Ki = 15.0 nM 7.82
CHEMBL233681 Ki = 19.0 nM 7.72
CHEMBL429440 Ki = 21.0 nM 7.68
CHEMBL232010 Ki = 25.0 nM 7.60