Assay Detail
Binding
CHEMBL902328
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Displacement of [125I]PYY from NPY1 receptor expressed in human SK-N-MC cells
17
Total Activities
17
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | SK-N-MC |
| Confidence | 9 — Direct single protein target |
| Curated By | Intermediate |
Publication
Identification of selective neuropeptide Y2 peptide agonists.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 17 | 7.01 | 7.68 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL439904 | — | — | 1 | 7.68 |
| CHEMBL269267 | — | — | 1 | 6.93 |
| CHEMBL238533 | — | — | 1 | 6.41 |
| CHEMBL397527 | — | — | 1 | - |
| CHEMBL392889 | — | — | 1 | - |
| CHEMBL268200 | — | — | 1 | - |
| CHEMBL227456 | — | — | 1 | - |
| CHEMBL429005 | — | — | 1 | - |
| CHEMBL397529 | — | — | 1 | - |
| CHEMBL411765 | — | — | 1 | - |
| CHEMBL266814 | — | — | 1 | - |
| CHEMBL436630 | — | — | 1 | - |
| CHEMBL437290 | — | — | 1 | - |
| CHEMBL397528 | — | — | 1 | - |
| CHEMBL241105 | — | — | 1 | - |
| CHEMBL411793 | — | — | 1 | - |
| CHEMBL411766 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL439904 | — | Ki | = | 21.0 | nM | 7.68 |
| CHEMBL269267 | — | Ki | = | 118.0 | nM | 6.93 |
| CHEMBL238533 | — | Ki | = | 390.0 | nM | 6.41 |
| CHEMBL397527 | — | Ki | > | 1000.0 | nM | - |
| CHEMBL392889 | — | Ki | > | 1000.0 | nM | - |
| CHEMBL268200 | — | Ki | > | 1000.0 | nM | - |
| CHEMBL227456 | — | Ki | > | 1000.0 | nM | - |
| CHEMBL429005 | — | Ki | > | 1000.0 | nM | - |
| CHEMBL397529 | — | Ki | > | 1000.0 | nM | - |
| CHEMBL411765 | — | Ki | > | 1000.0 | nM | - |
| CHEMBL266814 | — | Ki | > | 1000.0 | nM | - |
| CHEMBL436630 | — | Ki | > | 1000.0 | nM | - |
| CHEMBL437290 | — | Ki | > | 1000.0 | nM | - |
| CHEMBL397528 | — | Ki | > | 1000.0 | nM | - |
| CHEMBL241105 | — | Ki | > | 1000.0 | nM | - |
| CHEMBL411793 | — | Ki | > | 1000.0 | nM | - |
| CHEMBL411766 | — | Ki | > | 1000.0 | nM | - |