Assay Detail
Functional
CHEMBL925628
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Agonist activity at human recombinant FPRL1 expressed in CHO cells assessed as calcium flux by aequorin based bioluminescence assay
17
Total Activities
17
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | CHO |
| Confidence | 9 — Direct single protein target |
| Curated By | Intermediate |
Publication
New 'chemical probes' to examine the role of the hFPRL1 (or ALXR) receptor in inflammation.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 17 | 6.00 | 7.47 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL249132 | — | — | 1 | 7.47 |
| CHEMBL379761 | — | — | 1 | 7.36 |
| CHEMBL248928 | — | — | 1 | 6.89 |
| CHEMBL249742 | — | — | 1 | 6.57 |
| CHEMBL250347 | — | — | 1 | 6.16 |
| CHEMBL249537 | — | — | 1 | 6.09 |
| CHEMBL400089 | — | — | 1 | 6.08 |
| CHEMBL404003 | — | — | 1 | 5.99 |
| CHEMBL249338 | — | — | 1 | 5.83 |
| CHEMBL251772 | — | — | 1 | 5.82 |
| CHEMBL400723 | — | — | 1 | 5.73 |
| CHEMBL401313 | — | — | 1 | 5.57 |
| CHEMBL401314 | — | — | 1 | 5.46 |
| CHEMBL250143 | — | — | 1 | 5.29 |
| CHEMBL430016 | — | — | 1 | 4.91 |
| CHEMBL249339 | — | — | 1 | 4.85 |
| CHEMBL377169 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL249132 | — | EC50 | = | 34.0 | nM | 7.47 |
| CHEMBL379761 | — | EC50 | = | 44.0 | nM | 7.36 |
| CHEMBL248928 | — | EC50 | = | 130.0 | nM | 6.89 |
| CHEMBL249742 | — | EC50 | = | 270.0 | nM | 6.57 |
| CHEMBL250347 | — | EC50 | = | 690.0 | nM | 6.16 |
| CHEMBL249537 | — | EC50 | = | 810.0 | nM | 6.09 |
| CHEMBL400089 | — | EC50 | = | 830.0 | nM | 6.08 |
| CHEMBL404003 | — | EC50 | = | 1020.0 | nM | 5.99 |
| CHEMBL249338 | — | EC50 | = | 1490.0 | nM | 5.83 |
| CHEMBL251772 | — | EC50 | = | 1520.0 | nM | 5.82 |
| CHEMBL400723 | — | EC50 | = | 1870.0 | nM | 5.73 |
| CHEMBL401313 | — | EC50 | = | 2710.0 | nM | 5.57 |
| CHEMBL401314 | — | EC50 | = | 3500.0 | nM | 5.46 |
| CHEMBL250143 | — | EC50 | = | 5100.0 | nM | 5.29 |
| CHEMBL430016 | — | EC50 | = | 12200.0 | nM | 4.91 |
| CHEMBL249339 | — | EC50 | = | 14100.0 | nM | 4.85 |
| CHEMBL377169 | — | EC50 | > | 10000.0 | nM | - |