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Assay Detail

CHEMBL929419

Review assay metadata, readout intent, target linkage, and publication context from the same page.

ADMET
Inhibition of CYP3A4
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type ADMET
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

Cytochrome P450 3A4 (CHEMBL340)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Discovery and preclinical studies of 5-isopropyl-6-(5-methyl-1,3,4-oxadiazol-2-yl)-N-(2-methyl-1H-pyrrolo[2,3-b]pyridin-5-yl)pyrrolo[2,1-f][1,2,4]triazin-4-amine (BMS-645737), an in vivo active potent VEGFR-2 inhibitor.
Ruel R, Thibeault C, L'Heureux A, Martel A, Cai ZW, Wei D, Qian L, Barrish JC, Mathur A, D'Arienzo C, Hunt JT, Kamath A, Marathe P, Zhang Y, Derbin G, Wautlet B, Mortillo S, Jeyaseelan R, Henley B, Tejwani R, Bhide RS, Trainor GL, Fargnoli J, Lombardo LJ.
Bioorg Med Chem Lett (2008) 18 : 2985 -2989
PubMed 18395443 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 3 5.07 5.19

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL409442 1 5.19
CHEMBL261592 1 4.94
CHEMBL258694 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL409442 IC50 = 6400.0 nM 5.19
CHEMBL261592 IC50 = 11500.0 nM 4.94
CHEMBL258694 IC50 > 40000.0 nM -