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Assay Detail

CHEMBL978327

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Cytotoxicity against mouse P388 cells after 72 hrs by MTT method
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Mus musculus
Cell Type P388
Confidence 1 — Organism
Curated By Autocuration

Target

P388 (CHEMBL389)
Type CELL-LINE
Organism Mus musculus

Publication

10-Phenyl-[12]-cytochalasins Z7, Z8, and Z9 from the marine-derived fungus Spicaria elegans.
Liu R, Gu Q, Zhu W, Cui C, Fan G, Fang Y, Zhu T, Liu H.
J Nat Prod (2006) 69 : 871 -875
PubMed 16792402 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 5 4.69 7.03

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL494856 CYTOCHALASIN E 1 7.03
CHEMBL498454 1 4.25
CHEMBL497529 1 4.12
CHEMBL500120 CYTOCHALASIN K 1 4.05
CHEMBL498455 CYTOCHALASIN Z9 1 4.00

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL494856 CYTOCHALASIN E IC50 = 93.0 nM 7.03
CHEMBL498454 IC50 = 56000.0 nM 4.25
CHEMBL497529 IC50 = 75000.0 nM 4.12
CHEMBL500120 CYTOCHALASIN K IC50 = 89000.0 nM 4.05
CHEMBL498455 CYTOCHALASIN Z9 IC50 = 99000.0 nM 4.00