Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL991034

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against VZV Webster by plaque reduction assay
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Human alphaherpesvirus 3
Confidence 1 — Organism
Curated By Autocuration

Target

Human alphaherpesvirus 3 (CHEMBL613132)
Type ORGANISM
Organism Human alphaherpesvirus 3

Publication

Synthesis of 4-oxo-4,7-dihydrofuro[2,3-b]pyridine-5-carboxamides with broad-spectrum human herpesvirus polymerase inhibition.
Schnute ME, Brideau RJ, Collier SA, Cudahy MM, Hopkins TA, Knechtel ML, Oien NL, Sackett RS, Scott A, Stephan ML, Wathen MW, Wieber JL.
Bioorg Med Chem Lett (2008) 18 : 3856 -3859
PubMed 18595689 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 4 6.61 7.70

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL481172 1 7.70
CHEMBL479371 1 7.05
CHEMBL184 ACYCLOVIR 4.0 1 5.09
CHEMBL182 GANCICLOVIR 4.0 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL481172 IC50 = 20.0 nM 7.70
CHEMBL479371 IC50 = 90.0 nM 7.05
CHEMBL184 ACYCLOVIR IC50 = 8100.0 nM 5.09
CHEMBL182 GANCICLOVIR IC50 - -