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Assay Detail

CHEMBL995252

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antimicrobial activity against Escherichia coli CGMCC 1.2340
7
Total Activities
5
Compounds Tested
2
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Escherichia coli
Confidence 1 — Organism
Curated By Autocuration

Target

Escherichia coli (CHEMBL354)
Type ORGANISM
Organism Escherichia coli

Publication

Bioactive asterric acid derivatives from the Antarctic ascomycete fungus Geomyces sp.
Li Y, Sun B, Liu S, Jiang L, Liu X, Zhang H, Che Y.
J Nat Prod (2008) 71 : 1643 -1646
PubMed 18720971 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 5 5.44 5.98
MIC 2 - -

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL372795 STREPTOMYCIN 4.0 2 5.98
CHEMBL507180 GEOMYCIN C 2 4.89
CHEMBL499049 ETHYL ASTERRATE 1 -
CHEMBL501396 GEOMYCIN A 1 -
CHEMBL499873 BUTYL ASTERRATE 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL372795 STREPTOMYCIN IC50 = 1050.0 nM 5.98
CHEMBL507180 GEOMYCIN C IC50 = 12900.0 nM 4.89
CHEMBL507180 GEOMYCIN C MIC = 30300.0 nM -
CHEMBL372795 STREPTOMYCIN MIC = 11200.0 nM -
CHEMBL499049 ETHYL ASTERRATE IC50 > 50000.0 nM -
CHEMBL501396 GEOMYCIN A IC50 > 50000.0 nM -
CHEMBL499873 BUTYL ASTERRATE IC50 > 50000.0 nM -