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Assay Detail

CHEMBL996581

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antioxidant activity against cupric ion-induced lipid peroxidation in human LDL by TBA assay
10
Total Activities
10
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Confidence 1 — Organism
Curated By Autocuration

Publication

Isolation, identification, and antioxidant activity of three stilbene glucosides newly extracted from vitis vinifera cell cultures
Waffo Teguo P, Fauconneau B, Deffieux G, Huguet F, Vercauteren J, Merillon JM.
J Nat Prod (1998) 61 : 655 -657
PubMed 9599270 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 10 5.12 5.75

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL69863 PICEATANNOL 1 5.75
CHEMBL165 RESVERATROL 3.0 1 5.62
CHEMBL469920 Z-ASTRINGIN 1 5.60
CHEMBL358769 1 5.52
CHEMBL153 TROLOX 1 5.33
CHEMBL509386 Z-PICEID 1 4.78
CHEMBL87333 CIS-RESVERATROL 1 4.75
CHEMBL142652 PICEID 2.0 1 4.72
CHEMBL480100 E-RESVERATROLOSIDE 1 4.00
CHEMBL513583 Z-RESVERATROLOSIDE 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL69863 PICEATANNOL IC50 = 1800.0 nM 5.75
CHEMBL165 RESVERATROL IC50 = 2400.0 nM 5.62
CHEMBL469920 Z-ASTRINGIN IC50 = 2500.0 nM 5.60
CHEMBL358769 IC50 = 3000.0 nM 5.52
CHEMBL153 TROLOX IC50 = 4700.0 nM 5.33
CHEMBL509386 Z-PICEID IC50 = 16800.0 nM 4.78
CHEMBL87333 CIS-RESVERATROL IC50 = 18000.0 nM 4.75
CHEMBL142652 PICEID IC50 = 19100.0 nM 4.72
CHEMBL480100 E-RESVERATROLOSIDE IC50 = 100000.0 nM 4.00
CHEMBL513583 Z-RESVERATROLOSIDE IC50 = 150000.0 nM -