Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL997977

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against Vaccinia virus Copenhagen in HFF cells assessed as reduction of viral replication after 3 days
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Vaccinia virus
Cell Type HFF
Confidence 1 — Organism
Curated By Autocuration

Target

Vaccinia virus (CHEMBL613493)
Type ORGANISM
Organism Vaccinia virus

Publication

Effect of oral treatment with hexadecyloxypropyl-[(S)-9-(3-hydroxy-2- phosphonylmethoxypropyl)adenine] [(S)-HPMPA] or octadecyloxyethyl-(S)-HPMPA on cowpox or vaccinia virus infections in mice.
Quenelle DC, Collins DJ, Herrod BP, Keith KA, Trahan J, Beadle JR, Hostetler KY, Kern ER.
Antimicrob Agents Chemother (2007) 51 : 3940 -3947
PubMed 17846137 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 5 6.45 8.00

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL472584 1 8.00
CHEMBL487297 1 8.00
CHEMBL203321 BRINCIDOFOVIR 4.0 1 6.10
CHEMBL286534 1 5.57
CHEMBL5314375 CIDOFOVIR 4.0 1 4.58

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL472584 EC50 = 10.0 nM 8.00
CHEMBL487297 EC50 = 10.0 nM 8.00
CHEMBL203321 BRINCIDOFOVIR EC50 = 800.0 nM 6.10
CHEMBL286534 EC50 = 2700.0 nM 5.57
CHEMBL5314375 CIDOFOVIR EC50 = 26000.0 nM 4.58