Assay Detail
Binding
CHEMBL998565
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Inhibition of cFMS
13
Total Activities
13
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Intermediate |
Target
Macrophage colony-stimulating factor 1 receptor (CHEMBL1844) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Kinase array design, back to front: biaryl amides.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 13 | 6.72 | 8.40 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL521887 | — | — | 1 | 8.40 |
| CHEMBL497353 | — | — | 1 | 7.05 |
| CHEMBL496129 | — | — | 1 | 7.05 |
| CHEMBL497350 | — | — | 1 | 7.00 |
| CHEMBL526639 | — | — | 1 | 6.22 |
| CHEMBL523559 | — | — | 1 | 6.16 |
| CHEMBL485286 | — | — | 1 | 5.16 |
| CHEMBL485285 | — | — | 1 | - |
| CHEMBL495729 | — | — | 1 | - |
| CHEMBL497563 | — | — | 1 | - |
| CHEMBL522579 | — | — | 1 | - |
| CHEMBL521734 | — | — | 1 | - |
| CHEMBL478649 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL521887 | — | IC50 | = | 4.0 | nM | 8.40 |
| CHEMBL497353 | — | IC50 | = | 90.0 | nM | 7.05 |
| CHEMBL496129 | — | IC50 | = | 90.0 | nM | 7.05 |
| CHEMBL497350 | — | IC50 | = | 100.0 | nM | 7.00 |
| CHEMBL526639 | — | IC50 | = | 600.0 | nM | 6.22 |
| CHEMBL523559 | — | IC50 | = | 700.0 | nM | 6.16 |
| CHEMBL485286 | — | IC50 | = | 7000.0 | nM | 5.16 |
| CHEMBL485285 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL495729 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL497563 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL522579 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL521734 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL478649 | — | IC50 | > | 20000.0 | nM | - |