Assay Detail
ADMET
CHEMBL999263
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of human CYP3A4
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | ADMET |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Isolation of cytochrome P450 inhibitors from strawberry fruit, Fragaria ananassa.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 6.16 | 6.16 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL266564 | TILIROSIDE | — | 1 | 6.16 |
| CHEMBL499705 | — | — | 1 | 6.16 |
| CHEMBL484029 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL266564 | TILIROSIDE | IC50 | = | 700.0 | nM | 6.16 |
| CHEMBL499705 | — | IC50 | = | 700.0 | nM | 6.16 |
| CHEMBL484029 | — | IC50 | = | 120000.0 | nM | - |