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Compound Detail

CHEMBL113074

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COC[C@H]1O[C@@H](Oc2cc(/C=C/c3cc(OC)cc(OC)c3)ccc2OC)[C@H](OC)[C@@H](OC)[C@@H]1OC

Basic Information

ChEMBL ID CHEMBL113074
Phase Preclinical
Structure Type MOL
InChI Key SUCVNWYOBRSXKG-XWKSYUBDSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
1
Publications
0
Known Names

Molecular Properties

504.6
MW (Da)
3.68
ALogP
9
HBA
0
HBD
83.1
PSA (Ų)
0.40
QED
1
Ro5 Violations
12
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

Natural Product First in Class Prodrug

Extended Properties

Molecular Formula C27H36O9
MW 504.58
Aromatic Rings 2
Heavy Atoms 36
NP-Likeness 0.76

Activity Summary

IC50 1 meas. best 4.57

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Mus musculus
CHEMBL375
IC50 4.57 4.57 27000.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Mus musculus IC50 = 27000.0 nM 4.57 Inhibitory activity against nitric oxide production in LPS-activated mouse perit... 10714491

Literature References

PubMed DOI Target Context # Activities
10714491 10.1016/s0960-894x(99)00702-7 Mus musculus 1

Data from ChEMBL 36 via Core Engine