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Compound Detail

CHEMBL132535

GLYCYRIN
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COc1cc2oc(=O)c(-c3ccc(O)cc3O)cc2c(OC)c1CC=C(C)C

Basic Information

ChEMBL ID CHEMBL132535
Name GLYCYRIN
Phase Preclinical
Structure Type MOL
InChI Key FWWGXZYUURXJLK-UHFFFAOYSA-N
2
Targets
2
Activities
2
Assay Types
0
PK Parameters
11
Publications
0
Known Names

Molecular Properties

382.4
MW (Da)
4.40
ALogP
6
HBA
2
HBD
89.1
PSA (Ų)
0.50
QED
0
Ro5 Violations
5
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

Natural Product First in Class Prodrug

Extended Properties

Molecular Formula C22H22O6
MW 382.41
Aromatic Rings 3
Heavy Atoms 28
NP-Likeness 1.56

Activity Summary

EC50 1 meas. best 4.05
Ki 1 meas. best 4.37

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Unchecked
CHEMBL612545
Ki 4.37 4.37 42600.0 1
NON-PROTEIN TARGET
CHEMBL3879801
EC50 4.05 4.05 88100.0 1

Activity Data Samples

Top measurements by pChEMBL value

Literature References

PubMed DOI Target Context # Activities
28196701 10.1016/j.bmcl.2017.01.095 Unchecked 9
14643306 10.1016/j.bmcl.2003.09.052 Mus musculus 8
20850329 10.1016/j.bmc.2010.07.073 NON-PROTEIN TARGET 4
20064716 10.1016/j.bmcl.2009.12.106 Unchecked 2
20850329 10.1016/j.bmc.2010.07.073 ADMET 1
20850329 10.1016/j.bmc.2010.07.073 Unchecked 1
22074222 10.1021/np2004775 Streptococcus mutans 1
22074222 10.1021/np2004775 Streptococcus sobrinus 1
22074222 10.1021/np2004775 Prevotella intermedia 1
26841168 10.1021/acs.jnatprod.5b00877 Nuclear factor erythroid 2-related factor 2 1
28196701 10.1016/j.bmcl.2017.01.095 Bacillus subtilis 1

Data from ChEMBL 36 via Core Engine