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Compound Detail

CHEMBL1449136

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O=C1COc2ccc(-c3nnc(O)c4ccccc34)cc2N1

Basic Information

ChEMBL ID CHEMBL1449136
Phase Preclinical
Structure Type MOL
InChI Key AFSGHGHBHNFUDB-UHFFFAOYSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
0
Publications
0
Known Names

Molecular Properties

293.3
MW (Da)
2.33
ALogP
5
HBA
2
HBD
84.3
PSA (Ų)
0.72
QED
0
Ro5 Violations
1
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C16H11N3O3
MW 293.28
Aromatic Rings 3
Heavy Atoms 22
NP-Likeness -1.15

Activity Summary

IC50 1 meas. best 5.28

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
H9c2
CHEMBL614576
IC50 5.28 5.28 5261.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
H9c2 IC50 = 5261.0 nM 5.28 PUBCHEM_BIOASSAY: Dose response confirmation of uHTS hits for small molecule mod... -

Data from ChEMBL 36 via Core Engine