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Compound Detail

CHEMBL145868

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O=c1nc2oc(-c3ccc(Cl)cc3)cc2cn1[C@H]1C[C@H](O)[C@@H](CO)O1

Basic Information

ChEMBL ID CHEMBL145868
Phase Preclinical
Structure Type MOL
InChI Key RHYTZFFQLDUOIS-NWANDNLSSA-N
1
Targets
2
Activities
1
Assay Types
0
PK Parameters
2
Publications
0
Known Names

Molecular Properties

362.8
MW (Da)
1.95
ALogP
7
HBA
2
HBD
97.7
PSA (Ų)
0.74
QED
0
Ro5 Violations
3
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C17H15ClN2O5
MW 362.77
Aromatic Rings 3
Heavy Atoms 25
NP-Likeness 0.49

Activity Summary

EC50 2 meas. best 7.0

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Human alphaherpesvirus 3
CHEMBL613132
EC50 7.0 7.0 100.0 2

Activity Data Samples

Top measurements by pChEMBL value

Literature References

PubMed DOI Target Context # Activities
11150169 10.1021/jm000210m Human alphaherpesvirus 3 6
11150169 10.1021/jm000210m No relevant target 1

Data from ChEMBL 36 via Core Engine