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Compound Detail

CHEMBL1631222

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Nc1nc(=O)n([C@@H]2S[C@H](CO)[C@@H](O)[C@@H]2O)cc1F

Basic Information

ChEMBL ID CHEMBL1631222
Phase Preclinical
Structure Type MOL
InChI Key QDVOFRWTPUEFTR-MNCSTQPFSA-N
2
Targets
2
Activities
1
Assay Types
0
PK Parameters
3
Publications
0
Known Names

Molecular Properties

277.3
MW (Da)
-1.71
ALogP
8
HBA
4
HBD
121.6
PSA (Ų)
0.51
QED
0
Ro5 Violations
2
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C9H12FN3O4S
MW 277.28
Aromatic Rings 1
Heavy Atoms 18
NP-Likeness 0.12

Activity Summary

EC50 2 meas. best 7.0

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Vaccinia virus
CHEMBL613493
EC50 7.0 7.0 100.0 1
Cowpox virus
CHEMBL612672
EC50 6.4 6.4 400.0 1

Activity Data Samples

Top measurements by pChEMBL value

Literature References

PubMed DOI Target Context # Activities
19029322 10.1128/aac.01257-08 Vaccinia virus 4
19029322 10.1128/aac.01257-08 Cowpox virus 2
19029322 10.1128/aac.01257-08 HFF 2

Data from ChEMBL 36 via Core Engine