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Compound Detail

CHEMBL1824865

INFLATIN F
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COc1cc(=O)oc2c1[C@H](O[C@@H]1O[C@@H](C)[C@H](C)c3oc(=O)cc(OC)c31)O[C@@H](C)[C@@H]2C

Basic Information

ChEMBL ID CHEMBL1824865
Name INFLATIN F
Phase Preclinical
Structure Type MOL
InChI Key CGCDOVOCJQXOOK-NVXFIYROSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
6
Publications
0
Known Names

Molecular Properties

434.4
MW (Da)
3.37
ALogP
9
HBA
0
HBD
106.6
PSA (Ų)
0.72
QED
0
Ro5 Violations
4
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

Natural Product First in Class Prodrug

Extended Properties

Molecular Formula C22H26O9
MW 434.44
Aromatic Rings 2
Heavy Atoms 31
NP-Likeness 1.11

Activity Summary

IC50 1 meas. best 4.24

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
NON-PROTEIN TARGET
CHEMBL3879801
IC50 4.24 4.24 57500.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
NON-PROTEIN TARGET IC50 = 57500.0 nM 4.24 Cytotoxicity against human Hep3B2 cells after 72 hrs by MTS assay 21812410

Literature References

PubMed DOI Target Context # Activities
21812410 10.1021/np200431k NON-PROTEIN TARGET 4
21812410 10.1021/np200431k A549 1
21812410 10.1021/np200431k A-375 1
21812410 10.1021/np200431k MCF7 1
21812410 10.1021/np200431k PANC-1 1
21812410 10.1021/np200431k HaCaT 1

Data from ChEMBL 36 via Core Engine