Skip to main content
Free research Free research Free compound review with research home and workspace preview
Quick search ChEMBL 36
Compound Detail

CHEMBL2327013

Enter ChEMBL ID:
Free Research Context This compound will appear in recent viewed items on the research home for this browser.
Research home View demo workspace
Cc1ccc2c(Sc3cc(Cl)cc(Cl)c3)c(CCCC(N)=O)[nH]c2c1

Basic Information

ChEMBL ID CHEMBL2327013
Phase Preclinical
Structure Type MOL
InChI Key IXDGDLPUEYGBBL-UHFFFAOYSA-N
2
Targets
2
Activities
1
Assay Types
0
PK Parameters
3
Publications
0
Known Names

Molecular Properties

393.3
MW (Da)
5.74
ALogP
2
HBA
2
HBD
58.9
PSA (Ų)
0.56
QED
1
Ro5 Violations
6
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C19H18Cl2N2OS
MW 393.34
Aromatic Rings 3
Heavy Atoms 25
NP-Likeness -0.85

Activity Summary

IC50 2 meas. best 6.68

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Uracil-DNA glycosylase
CHEMBL3988595
IC50 6.68 6.68 208.0 1
Vaccinia virus
CHEMBL613493
IC50 6.68 6.68 208.0 1

Activity Data Samples

Top measurements by pChEMBL value

Literature References

PubMed DOI Target Context # Activities
23527789 10.1021/jm301735k Unchecked 1
23527789 10.1021/jm301735k Vaccinia virus 1
23527789 10.1021/jm301735k BSC-1 1

Data from ChEMBL 36 via Core Engine