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Compound Detail

CHEMBL233207

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CN(NS(C)(=O)=O)c1nc(N)nc2c1ncn2[C@@H]1O[C@@H]2OP(=O)(OCCSC(=O)C(C)(C)C)O[C@H]2[C@@]1(C)O

Basic Information

ChEMBL ID CHEMBL233207
Phase Preclinical
Structure Type MOL
InChI Key VYUQSXGWJYQADG-HICYRPCPSA-N
2
Targets
2
Activities
1
Assay Types
0
PK Parameters
2
Publications
0
Known Names

Molecular Properties

595.6
MW (Da)
0.76
ALogP
16
HBA
3
HBD
210.3
PSA (Ų)
0.22
QED
2
Ro5 Violations
8
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C19H30N7O9PS2
MW 595.60
Aromatic Rings 2
Heavy Atoms 38
NP-Likeness -0.02

Activity Summary

EC50 2 meas. best 7.66

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Hepatitis C virus
CHEMBL379
EC50 7.66 7.66 22.0 1
Bovine viral diarrhea virus 1
CHEMBL612571
EC50 7.48 7.48 33.0 1

Activity Data Samples

Top measurements by pChEMBL value

Literature References

PubMed DOI Target Context # Activities
17331721 10.1016/j.bmcl.2007.02.030 Hepatitis C virus 1
17331721 10.1016/j.bmcl.2007.02.030 Bovine viral diarrhea virus 1 1

Data from ChEMBL 36 via Core Engine