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Compound Detail

CHEMBL234888

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C[C@H]1C=C(C[C@H](O)CCCCCCCCCC[C@@H](O)[C@H]2CC[C@H]([C@H]3CC[C@H]([C@H](O)CCCCCCCCCCCO)O3)O2)C(=O)O1

Basic Information

ChEMBL ID CHEMBL234888
Phase Preclinical
Structure Type MOL
InChI Key YHBCAVBRJLHDIC-QTUSKHGGSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
1
Publications
0
Known Names

Molecular Properties

653.0
MW (Da)
7.22
ALogP
8
HBA
4
HBD
125.7
PSA (Ų)
0.05
QED
2
Ro5 Violations
27
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C38H68O8
MW 652.95
Aromatic Rings 0
Heavy Atoms 46
NP-Likeness 1.81

Activity Summary

IC50 1 meas. best 9.22

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
HCT-116
CHEMBL394
IC50 9.22 9.22 0.6 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
HCT-116 IC50 = 0.6 nM 9.22 Cytotoxicity against HCT116 cells 17329102

Literature References

PubMed DOI Target Context # Activities
17329102 10.1016/j.bmcl.2007.02.033 HCT-116 1

Data from ChEMBL 36 via Core Engine