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Compound Detail

CHEMBL3115425

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O=[N+]([O-])c1ccc2nc3c(c(-c4ccccc4)c2c1)CCCCC3

Basic Information

ChEMBL ID CHEMBL3115425
Phase Preclinical
Structure Type MOL
InChI Key LIXPGQKGCDZBRO-UHFFFAOYSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
2
Publications
0
Known Names

Molecular Properties

318.4
MW (Da)
5.08
ALogP
3
HBA
0
HBD
56.0
PSA (Ų)
0.38
QED
1
Ro5 Violations
2
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C20H18N2O2
MW 318.38
Aromatic Rings 3
Heavy Atoms 24
NP-Likeness -1.00

Activity Summary

IC50 1 meas. best 4.21

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Mycobacterium tuberculosis
CHEMBL360
IC50 4.21 4.21 61930.0 1

Activity Data Samples

Top measurements by pChEMBL value

Literature References

PubMed DOI Target Context # Activities
24412719 10.1016/j.ejmech.2013.12.013 Mycobacterium tuberculosis 15
24412719 10.1016/j.ejmech.2013.12.013 J774 3

Data from ChEMBL 36 via Core Engine