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Compound Detail

CHEMBL3138693

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CC(=O)O[C@@H]1C[C@H]2C(C)(C)[C@@H](O)CC[C@]2(C)[C@H]2CC[C@]3(C)C(=CC(=O)O[C@H]3c3ccoc3)[C@@]21C

Basic Information

ChEMBL ID CHEMBL3138693
Phase Preclinical
Structure Type MOL
InChI Key FJIIOEQLAAKWEL-VSELDIKBSA-N
2
Targets
4
Activities
1
Assay Types
0
PK Parameters
2
Publications
0
Known Names

Molecular Properties

470.6
MW (Da)
5.37
ALogP
6
HBA
1
HBD
86.0
PSA (Ų)
0.59
QED
1
Ro5 Violations
2
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

Natural Product First in Class Prodrug

Extended Properties

Molecular Formula C28H38O6
MW 470.61
Aromatic Rings 1
Heavy Atoms 34
NP-Likeness 3.31

Activity Summary

Ki 4 meas. best 6.03

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Solute carrier organic anion transporter family member 1B1
CHEMBL1697668
Ki 6.03 5.93 930.0 2
Solute carrier organic anion transporter family member 1B3
CHEMBL1743121
Ki 5.62 5.61 2390.0 2

Activity Data Samples

Top measurements by pChEMBL value

Literature References

PubMed DOI Target Context # Activities
23571415 10.1124/mol.112.084152 Solute carrier organic anion transporter family member 1B3 3
23571415 10.1124/mol.112.084152 Solute carrier organic anion transporter family member 1B1 3

Data from ChEMBL 36 via Core Engine