Skip to main content
Free research Free research Free compound review with research home and workspace preview
Quick search ChEMBL 36
Compound Detail

CHEMBL3143164

Enter ChEMBL ID:
Free Research Context This compound will appear in recent viewed items on the research home for this browser.
Research home View demo workspace
CCCCCCCCCCCCc1cc2cn([C@H]3C[C@H](O)[C@@H](CO)O3)c(=O)nc2o1

Basic Information

ChEMBL ID CHEMBL3143164
Phase Preclinical
Structure Type MOL
InChI Key TVRKQWFWACVJGU-PWRODBHTSA-N
1
Targets
2
Activities
1
Assay Types
0
PK Parameters
2
Publications
0
Known Names

Molecular Properties

420.6
MW (Da)
4.09
ALogP
7
HBA
2
HBD
97.7
PSA (Ų)
0.47
QED
0
Ro5 Violations
13
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C23H36N2O5
MW 420.55
Aromatic Rings 2
Heavy Atoms 30
NP-Likeness 0.78

Activity Summary

EC50 2 meas. best 5.96

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Human alphaherpesvirus 3
CHEMBL613132
EC50 5.96 5.925 1100.0 2

Activity Data Samples

Top measurements by pChEMBL value

Literature References

PubMed DOI Target Context # Activities
10579812 10.1021/jm990346o Human alphaherpesvirus 3 4
10579812 10.1021/jm990346o HEL 2

Data from ChEMBL 36 via Core Engine