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Compound Detail

CHEMBL3143183

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O=c1[nH]c(=O)n([C@H]2C[C@H](O)[C@@H](CO)O2)cc1C#CCCCCCCCCCF

Basic Information

ChEMBL ID CHEMBL3143183
Phase Preclinical
Structure Type MOL
InChI Key LGIBDFUFZFWHIM-RCCFBDPRSA-N
1
Targets
4
Activities
1
Assay Types
0
PK Parameters
3
Publications
0
Known Names

Molecular Properties

396.5
MW (Da)
1.62
ALogP
6
HBA
3
HBD
104.5
PSA (Ų)
0.41
QED
0
Ro5 Violations
10
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C20H29FN2O5
MW 396.46
Aromatic Rings 1
Heavy Atoms 28
NP-Likeness 0.59

Activity Summary

EC50 4 meas. best 4.66

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Human alphaherpesvirus 3
CHEMBL613132
EC50 4.66 4.59 22000.0 4

Activity Data Samples

Top measurements by pChEMBL value

Literature References

PubMed DOI Target Context # Activities
10866384 10.1016/s0960-894x(00)00193-1 Human alphaherpesvirus 3 4
10866384 10.1016/s0960-894x(00)00193-1 NON-PROTEIN TARGET 1
10866384 10.1016/s0960-894x(00)00193-1 HEL 1

Data from ChEMBL 36 via Core Engine