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Compound Detail

CHEMBL3331395

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N#CCn1cc(CN(C2=CC(=O)c3ccccc3C2=O)c2ccccc2)nn1

Basic Information

ChEMBL ID CHEMBL3331395
Phase Preclinical
Structure Type MOL
InChI Key QRWXWGZOWNIKQL-UHFFFAOYSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
1
Publications
0
Known Names

Molecular Properties

369.4
MW (Da)
2.77
ALogP
7
HBA
0
HBD
91.9
PSA (Ų)
0.69
QED
0
Ro5 Violations
5
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C21H15N5O2
MW 369.38
Aromatic Rings 3
Heavy Atoms 28
NP-Likeness -0.74

Activity Summary

IC50 1 meas. best 5.0

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Mycobacterium tuberculosis
CHEMBL360
IC50 5.0 5.0 9950.0 1

Activity Data Samples

Top measurements by pChEMBL value

Literature References

PubMed DOI Target Context # Activities
25129868 10.1016/j.ejmech.2014.08.009 Mycobacterium tuberculosis 3

Data from ChEMBL 36 via Core Engine