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Compound Detail

CHEMBL34246

IPROZILAMINE
🧪 Phase II
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🧪 Phase II
CSc1c(Cl)nc(NC(C)C)nc1N1CCN(C)CC1

Basic Information

ChEMBL ID CHEMBL34246
Name IPROZILAMINE
Phase Phase II
Structure Type MOL
InChI Key UMMYPDFDLDVDCZ-UHFFFAOYSA-N

Known Names

Iprozilamina Iprozilamine
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
1
Publications
2
Known Names

Molecular Properties

315.9
MW (Da)
2.42
ALogP
6
HBA
1
HBD
44.3
PSA (Ų)
0.68
QED
0
Ro5 Violations
4
Rot. Bonds

Drug Information

Molecule Type Small molecule
Chirality Achiral

Extended Properties

Molecular Formula C13H22ClN5S
MW 315.87
Aromatic Rings 1
Heavy Atoms 20
NP-Likeness -1.16

Activity Summary

Ki 1 meas. best 5.1

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Dopamine receptor
CHEMBL2093868
Ki 5.1 5.1 8000.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Dopamine receptor Ki = 8000.0 nM 5.1 In vitro ability to displace [3H]spiroperidol from rat dopamine receptor 7154006

Literature References

PubMed DOI Target Context # Activities
7154006 10.1021/jm00354a014 Dopamine receptor 1

Data from ChEMBL 36 via Core Engine