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Compound Detail

CHEMBL3633915

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Oc1ccc(C2=Cc3cc(CN4CCOCC4)c(O)cc3OC2)cc1

Basic Information

ChEMBL ID CHEMBL3633915
Phase Preclinical
Structure Type MOL
InChI Key BLWWOZKIALMCCY-UHFFFAOYSA-N
1
Targets
2
Activities
1
Assay Types
0
PK Parameters
2
Publications
0
Known Names

Molecular Properties

339.4
MW (Da)
2.86
ALogP
5
HBA
2
HBD
62.2
PSA (Ų)
0.90
QED
0
Ro5 Violations
3
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C20H21NO4
MW 339.39
Aromatic Rings 2
Heavy Atoms 25
NP-Likeness 0.12

Activity Summary

IC50 2 meas. best 4.06

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
NON-PROTEIN TARGET
CHEMBL3879801
IC50 4.06 4.06 86800.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
NON-PROTEIN TARGET IC50 = 86800.0 nM 4.06 Antiproliferative effects against human SHEP cells after 72 hrs by Alamar blue a... 26432036

Literature References

PubMed DOI Target Context # Activities
26432036 10.1016/j.bmcl.2015.09.027 MDA-MB-231 1
26432036 10.1016/j.bmcl.2015.09.027 NON-PROTEIN TARGET 1

Data from ChEMBL 36 via Core Engine