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Compound Detail

CHEMBL3746578

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O=C(OCCOC12CC3CC(CC(C3)C1)C2)c1cc(N(O)C2CCCO2)on1

Basic Information

ChEMBL ID CHEMBL3746578
Phase Preclinical
Structure Type MOL
InChI Key ZZEQQLFUXTXKIT-UHFFFAOYSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
5
Publications
0
Known Names

Molecular Properties

392.4
MW (Da)
3.15
ALogP
8
HBA
1
HBD
94.3
PSA (Ų)
0.43
QED
0
Ro5 Violations
7
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C20H28N2O6
MW 392.45
Aromatic Rings 1
Heavy Atoms 28
NP-Likeness -0.50

Activity Summary

IC50 1 meas. best 4.46

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Brain
CHEMBL613617
IC50 4.46 4.46 35000.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Brain IC50 = 35000.0 nM 4.46 Antioxidant activity in albino rat brain homogenate assessed as inhibition of Fe... 26753816

Literature References

PubMed DOI Target Context # Activities
26753816 10.1016/j.bmc.2015.12.040 Unchecked 5
26753816 10.1016/j.bmc.2015.12.040 Brain 2
26753816 10.1016/j.bmc.2015.12.040 Seed linoleate 13S-lipoxygenase-1 1
26753816 10.1016/j.bmc.2015.12.040 No relevant target 1
26753816 10.1016/j.bmc.2015.12.040 ADMET 1

Data from ChEMBL 36 via Core Engine