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Compound Detail

CHEMBL3926548

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CC1(C)OC[C@@]2(C[C@@]34CC[C@H]5C(C)(C)C(=O)CC[C@]5(C)[C@H]3CC[C@H]2C4)O1

Basic Information

ChEMBL ID CHEMBL3926548
Phase Preclinical
Structure Type MOL
InChI Key CUMXMFWUFRFNQK-OCIMHDLJSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
1
Publications
0
Known Names

Molecular Properties

360.5
MW (Da)
5.12
ALogP
3
HBA
0
HBD
35.5
PSA (Ų)
0.60
QED
1
Ro5 Violations
0
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

Natural Product First in Class Prodrug

Extended Properties

Molecular Formula C23H36O3
MW 360.54
Aromatic Rings 0
Heavy Atoms 26
NP-Likeness 3.33

Activity Summary

IC50 1 meas. best 5.09

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
NON-PROTEIN TARGET
CHEMBL3879801
IC50 5.09 5.09 8146.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
NON-PROTEIN TARGET IC50 = 8146.0 nM 5.09 Cytotoxicity against human Hep3B cells assessed as cell growth inhibition by MTT... 27913179

Literature References

PubMed DOI Target Context # Activities
27913179 10.1016/j.bmcl.2016.11.063 NON-PROTEIN TARGET 2

Data from ChEMBL 36 via Core Engine