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Compound Detail

CHEMBL397573

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CCCOCC(C)(C)C(=O)SCCOP1(=O)O[C@H]2O[C@@H](n3cnc4c(N(C)NS(C)(=O)=O)ncnc43)[C@](C)(O)[C@@H]2O1

Basic Information

ChEMBL ID CHEMBL397573
Phase Preclinical
Structure Type MOL
InChI Key ZHJFHFHGYJYCTJ-KLOPIGLZSA-N
2
Targets
2
Activities
1
Assay Types
0
PK Parameters
2
Publications
0
Known Names

Molecular Properties

638.7
MW (Da)
1.59
ALogP
16
HBA
2
HBD
193.5
PSA (Ų)
0.18
QED
2
Ro5 Violations
13
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C22H35N6O10PS2
MW 638.66
Aromatic Rings 2
Heavy Atoms 41
NP-Likeness -0.08

Activity Summary

EC50 2 meas. best 7.41

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Hepatitis C virus
CHEMBL379
EC50 7.41 7.41 39.0 1
Bovine viral diarrhea virus 1
CHEMBL612571
EC50 6.96 6.96 110.0 1

Activity Data Samples

Top measurements by pChEMBL value

Literature References

PubMed DOI Target Context # Activities
17331721 10.1016/j.bmcl.2007.02.030 Hepatitis C virus 1
17331721 10.1016/j.bmcl.2007.02.030 Bovine viral diarrhea virus 1 1

Data from ChEMBL 36 via Core Engine