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Compound Detail

CHEMBL448034

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C[C@H]1[C@H](O[C@H]2O[C@@H]3O[C@]4(C)CC[C@H]5[C@H](C)CC[C@@H]([C@H]2C)[C@@]35O4)O[C@@H]2O[C@]3(C)CC[C@H]4[C@H](C)CC[C@@H]1[C@@]24O3

Basic Information

ChEMBL ID CHEMBL448034
Phase Preclinical
Structure Type MOL
InChI Key KQEOZJHTBAWJLC-AZVVYKQTSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
1
Publications
0
Known Names

Molecular Properties

518.7
MW (Da)
5.56
ALogP
7
HBA
0
HBD
64.6
PSA (Ų)
0.47
QED
2
Ro5 Violations
2
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C30H46O7
MW 518.69
Aromatic Rings 0
Heavy Atoms 37
NP-Likeness 2.02

Activity Summary

IC50 1 meas. best 5.05

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
NON-PROTEIN TARGET
CHEMBL3879801
IC50 5.05 5.05 8900.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
NON-PROTEIN TARGET IC50 = 8900.0 nM 5.05 Cytotoxicity against mouse EN2 cells after 72 hrs by MTT assay 9134741

Literature References

PubMed DOI Target Context # Activities
9134741 10.1021/np9605495 NON-PROTEIN TARGET 1

Data from ChEMBL 36 via Core Engine