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Compound Detail

CHEMBL4534700

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NCCc1nc(-c2ccccn2)cs1

Basic Information

ChEMBL ID CHEMBL4534700
Phase Preclinical
Structure Type MOL
InChI Key STIRJTZFRKEHMZ-UHFFFAOYSA-N
1
Targets
2
Activities
1
Assay Types
0
PK Parameters
3
Publications
0
Known Names

Molecular Properties

205.3
MW (Da)
1.71
ALogP
4
HBA
1
HBD
51.8
PSA (Ų)
0.83
QED
0
Ro5 Violations
3
Rot. Bonds

Drug Information

Molecule Type Unknown
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C10H11N3S
MW 205.29
Aromatic Rings 2
Heavy Atoms 14
NP-Likeness -1.63

Activity Summary

IC50 2 meas. best 5.94

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Unchecked
CHEMBL612545
IC50 5.94 5.755 1158.3 2

Activity Data Samples

Top measurements by pChEMBL value

Literature References

PubMed DOI Target Context # Activities
- 10.6019/CHEMBL3988442 Unchecked 5
- 10.6019/CHEMBL4513160 Pseudomonas aeruginosa 2
- 10.6019/CHEMBL4513160 Acinetobacter baumannii 1

Data from ChEMBL 36 via Core Engine