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Compound Detail

CHEMBL4646622

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Cc1cc(C)c(CN2CCN(C(=S)SCc3nc4ccccc4s3)CC2)c(C)c1

Basic Information

ChEMBL ID CHEMBL4646622
Phase Preclinical
Structure Type MOL
InChI Key DKTISHMOHAYPAB-UHFFFAOYSA-N
1
Targets
2
Activities
1
Assay Types
0
PK Parameters
2
Publications
0
Known Names

Molecular Properties

441.7
MW (Da)
5.56
ALogP
5
HBA
0
HBD
19.4
PSA (Ų)
0.49
QED
1
Ro5 Violations
4
Rot. Bonds

Drug Information

Molecule Type Unknown
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C23H27N3S3
MW 441.69
Aromatic Rings 3
Heavy Atoms 29
NP-Likeness -1.84

Activity Summary

EC50 2 meas. best 4.69

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Human orthopneumovirus
CHEMBL613127
EC50 4.69 4.535 20600.0 2

Activity Data Samples

Top measurements by pChEMBL value

Literature References

PubMed DOI Target Context # Activities
32143992 10.1016/j.bmc.2020.115401 Human orthopneumovirus 2
32143992 10.1016/j.bmc.2020.115401 HEp-2 1

Data from ChEMBL 36 via Core Engine