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Compound Detail

CHEMBL466369

HORMOTHAMNIONE DIACETATE
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COc1c(OC)c(O)c2c(=O)c(C)c(/C=C/c3cc(OC(C)=O)cc(OC(C)=O)c3)oc2c1OC

Basic Information

ChEMBL ID CHEMBL466369
Name HORMOTHAMNIONE DIACETATE
Phase Preclinical
Structure Type MOL
InChI Key XDNKUKQCGIZSCU-BQYQJAHWSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
2
Publications
0
Known Names

Molecular Properties

484.5
MW (Da)
3.85
ALogP
10
HBA
1
HBD
130.7
PSA (Ų)
0.39
QED
0
Ro5 Violations
7
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C25H24O10
MW 484.46
Aromatic Rings 3
Heavy Atoms 35
NP-Likeness 1.07

Activity Summary

IC50 1 meas. best 4.74

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
HL-60
CHEMBL383
IC50 4.74 4.74 18300.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
HL-60 IC50 = 18300.0 nM 4.74 Antioxidant activity against TPA-induced ROS production in human HL60 cells by 2... 12762791

Literature References

PubMed DOI Target Context # Activities
12762791 10.1021/np0204038 HL-60 1
12762791 10.1021/np0204038 Radical scavenging activity 1

Data from ChEMBL 36 via Core Engine