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Compound Detail

CHEMBL467503

AMINODIPHENYLMETHANE
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NC(c1ccccc1)c1ccccc1

Basic Information

ChEMBL ID CHEMBL467503
Name AMINODIPHENYLMETHANE
Phase Preclinical
Structure Type MOL
InChI Key MGHPNCMVUAKAIE-UHFFFAOYSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
2
Publications
0
Known Names

Molecular Properties

183.2
MW (Da)
2.73
ALogP
1
HBA
1
HBD
26.0
PSA (Ų)
0.76
QED
0
Ro5 Violations
2
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C13H13N
MW 183.25
Aromatic Rings 2
Heavy Atoms 14
NP-Likeness -0.21

Activity Summary

Ki 1 meas. best 4.19

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Glutamate NMDA receptor
CHEMBL1907608
Ki 4.19 4.19 64000.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Glutamate NMDA receptor Ki = 64000.0 nM 4.19 Displacement of [3H]MK801 from NMDA receptor in rat brain neuronal membrane 19345586

Literature References

PubMed DOI Target Context # Activities
19345586 10.1016/j.bmc.2009.03.025 Glutamate NMDA receptor 2
26810833 10.1016/j.bmc.2015.12.036 Mycobacterium tuberculosis 1

Data from ChEMBL 36 via Core Engine