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Compound Detail

CHEMBL4796023

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CCCCCCCCn1c2ccc(C(C)=O)cc2c2cc(C(=O)/C=C/c3ccc(Cl)cc3)ccc21

Basic Information

ChEMBL ID CHEMBL4796023
Phase Preclinical
Structure Type MOL
InChI Key AVWRRVUHLBRJHW-WOJGMQOQSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
1
Publications
0
Known Names

Molecular Properties

486.1
MW (Da)
8.91
ALogP
3
HBA
0
HBD
39.1
PSA (Ų)
0.12
QED
1
Ro5 Violations
11
Rot. Bonds

Drug Information

Molecule Type Unknown
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C31H32ClNO2
MW 486.06
Aromatic Rings 4
Heavy Atoms 35
NP-Likeness -0.43

Activity Summary

IC50 1 meas. best 4.61

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Urease
CHEMBL4161
IC50 4.61 4.61 24680.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Urease IC50 = 24680.0 nM 4.61 Inhibition of jack bean urease assessed as reduction in ammonia production using... 31623971

Literature References

PubMed DOI Target Context # Activities
31623971 10.1016/j.bmc.2019.115123 Urease 2

Data from ChEMBL 36 via Core Engine