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Compound Detail

CHEMBL483601

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CC1=C2C[C@H]3[C@@H](CCC4=CC(=O)CC[C@@]43C)[C@@H]2CC[C@@]2(C1)O[C@@H]1C[C@H](C)CN(C)[C@H]1[C@H]2C

Basic Information

ChEMBL ID CHEMBL483601
Phase Preclinical
Structure Type MOL
InChI Key MWLZYTHDYNEXEN-CXHJXZPGSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
1
Publications
0
Known Names

Molecular Properties

437.7
MW (Da)
5.94
ALogP
3
HBA
0
HBD
29.5
PSA (Ų)
0.44
QED
1
Ro5 Violations
0
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C29H43NO2
MW 437.67
Aromatic Rings 0
Heavy Atoms 32
NP-Likeness 2.11

Activity Summary

EC50 1 meas. best 6.4

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Molecular identity unknown
CHEMBL612546
EC50 6.4 6.4 400.0 1

Activity Data Samples

Top measurements by pChEMBL value

Literature References

PubMed DOI Target Context # Activities
18842035 10.1021/jm8008508 Molecular identity unknown 1

Data from ChEMBL 36 via Core Engine