Skip to main content
Free research Free research Free compound review with research home and workspace preview
Quick search ChEMBL 36
Compound Detail

CHEMBL508096

Enter ChEMBL ID:
Free Research Context This compound will appear in recent viewed items on the research home for this browser.
Research home View demo workspace
C[C@H]1[C@@H](CCOP(C)(=O)OCC[C@H]2O[C@@H]3O[C@@]4(C)CC[C@H]5[C@H](C)CC[C@@H]([C@H]2C)[C@@]35O4)O[C@@H]2O[C@@]3(C)CC[C@H]4[C@H](C)CC[C@@H]1[C@@]24O3

Basic Information

ChEMBL ID CHEMBL508096
Phase Preclinical
Structure Type MOL
InChI Key TYVHFKHDAYFVJF-XVCDAZLWSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
2
Publications
0
Known Names

Molecular Properties

652.8
MW (Da)
7.26
ALogP
9
HBA
0
HBD
90.9
PSA (Ų)
0.25
QED
2
Ro5 Violations
8
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C35H57O9P
MW 652.81
Aromatic Rings 0
Heavy Atoms 45
NP-Likeness 1.46

Activity Summary

IC50 1 meas. best 4.55

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
HL-60
CHEMBL383
IC50 4.55 4.55 28140.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
HL-60 IC50 = 28140.0 nM 4.55 Anticancer activity against human HL60 cells by MTT assay 19136263

Literature References

PubMed DOI Target Context # Activities
19136263 10.1016/j.bmc.2008.12.017 HL-60 1
19136263 10.1016/j.bmc.2008.12.017 Plasmodium falciparum 1

Data from ChEMBL 36 via Core Engine