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Compound Detail

CHEMBL522168

PESTALOFONE C
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C=C(C)/C=C1C(=C2\C[C@H](O)[C@@H]3O[C@]3(CC=C(C)C)C2=O)/C=C(C)C[C@@]/12C[C@H](O)[C@@H]1O[C@]1(CC=C(C)C)C2=O

Basic Information

ChEMBL ID CHEMBL522168
Name PESTALOFONE C
Phase Preclinical
Structure Type MOL
InChI Key LJTKUBXRWULZKS-PDIAYQMFSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
1
Publications
0
Known Names

Molecular Properties

520.7
MW (Da)
4.78
ALogP
6
HBA
2
HBD
99.7
PSA (Ų)
0.31
QED
1
Ro5 Violations
5
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

Natural Product First in Class Prodrug

Extended Properties

Molecular Formula C32H40O6
MW 520.67
Aromatic Rings 0
Heavy Atoms 38
NP-Likeness 1.87

Activity Summary

IC50 1 meas. best 5.96

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Aspergillus fumigatus
CHEMBL363
IC50 5.96 5.96 1100.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Aspergillus fumigatus IC50 = 1100.0 nM 5.96 Antimicrobial activity against Aspergillus fumigatus ATCC 10894 19101157

Literature References

PubMed DOI Target Context # Activities
19101157 10.1016/j.bmc.2008.11.066 Aspergillus fumigatus 2

Data from ChEMBL 36 via Core Engine