Skip to main content
Free research Free research Free compound review with research home and workspace preview
Quick search ChEMBL 36
Compound Detail

CHEMBL5283434

Enter ChEMBL ID:
Free Research Context This compound will appear in recent viewed items on the research home for this browser.
Research home View demo workspace
CCCCCCCCCCCCCCCCCCC/C=C/C(=O)OC[C@H](CO[C@@H]1O[C@H](CO[C@H]2O[C@H](CO)[C@H](O)[C@H](O)[C@H]2O)[C@H](O)[C@H](O)[C@H]1O)OC(=O)CCCCCCCCCCCCCCCCCCC

Basic Information

ChEMBL ID CHEMBL5283434
Phase Preclinical
Structure Type MOL
InChI Key FPBOHGQTFPCPBD-WIGFTALISA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
1
Publications
0
Known Names

Molecular Properties

1031.5
MW (Da)

Drug Information

Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C57H106O15
MW 1031.46

Activity Summary

IC50 1 meas. best 4.81

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Fatty acid synthase
CHEMBL1795136
IC50 4.81 4.81 15600.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Fatty acid synthase IC50 = 15600.0 nM 4.81 Inhibition of Fatty acid synthase in chicken liver using [3H]-acetyl CoA as subs... 29126728

Literature References

PubMed DOI Target Context # Activities
29126728 10.1016/j.ejmech.2017.10.015 Fatty acid synthase 1

Data from ChEMBL 36 via Core Engine