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Compound Detail

CHEMBL5604846

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O=C(Nc1cc(Cl)cc(-c2ccc3[nH]nc(C(=O)O)c3c2)c1)OCc1ccccc1

Basic Information

ChEMBL ID CHEMBL5604846
Phase Preclinical
Structure Type MOL
InChI Key HGXOIZSZLJEXKS-UHFFFAOYSA-N
2
Targets
4
Activities
1
Assay Types
0
PK Parameters
5
Publications
0
Known Names

Molecular Properties

421.8
MW (Da)
5.33
ALogP
4
HBA
3
HBD
104.3
PSA (Ų)
0.40
QED
1
Ro5 Violations
5
Rot. Bonds

Drug Information

Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C22H16ClN3O4
MW 421.84
Aromatic Rings 4
Heavy Atoms 30
NP-Likeness -1.25

Activity Summary

IC50 4 meas. best 5.3

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Genome polyprotein
CHEMBL5980
IC50 5.3 5.18 5003.0 3
Nonstructural protein 3
CHEMBL4523954
IC50 4.75 4.75 17836.0 1

Activity Data Samples

Top measurements by pChEMBL value

Literature References

PubMed DOI Target Context # Activities
- 10.6019/CHEMBL5604063 Genome polyprotein 3
- 10.6019/CHEMBL5661943 Zika virus 2
- 10.6019/CHEMBL5661943 dengue virus type 2 2
- 10.6019/CHEMBL5661955 ADMET 2
- 10.6019/CHEMBL5604062 Nonstructural protein 3 1

Data from ChEMBL 36 via Core Engine