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Compound Detail

CHEMBL5606200

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CCc1cc(C(=O)Nc2cccc(-c3nnn[nH]3)c2)sc1-c1ccc(Cl)cc1

Basic Information

ChEMBL ID CHEMBL5606200
Phase Preclinical
Structure Type MOL
InChI Key GTLKUZJXLRRDRT-UHFFFAOYSA-N
2
Targets
4
Activities
1
Assay Types
0
PK Parameters
5
Publications
0
Known Names

Molecular Properties

409.9
MW (Da)
5.06
ALogP
5
HBA
2
HBD
83.6
PSA (Ų)
0.48
QED
1
Ro5 Violations
5
Rot. Bonds

Drug Information

Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C20H16ClN5OS
MW 409.90
Aromatic Rings 4
Heavy Atoms 28
NP-Likeness -2.09

Activity Summary

IC50 4 meas. best 5.25

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Genome polyprotein
CHEMBL5980
IC50 5.25 5.235 5661.0 2
Nonstructural protein 3
CHEMBL4523954
IC50 4.93 4.855 11802.0 2

Activity Data Samples

Top measurements by pChEMBL value

Literature References

PubMed DOI Target Context # Activities
- 10.6019/CHEMBL5661943 Zika virus 4
- 10.6019/CHEMBL5661943 dengue virus type 2 4
- 10.6019/CHEMBL5661955 ADMET 4
- 10.6019/CHEMBL5604063 Genome polyprotein 3
- 10.6019/CHEMBL5604062 Nonstructural protein 3 2

Data from ChEMBL 36 via Core Engine