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Compound Detail

CHEMBL5647387

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CCOc1ccc2nc(NCCOC)nc(Nc3cc(C(F)(F)F)cc(C(F)(F)F)c3)c2c1

Basic Information

ChEMBL ID CHEMBL5647387
Phase Preclinical
Structure Type MOL
InChI Key BTRZCKSFGDPKNU-UHFFFAOYSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
3
Publications
0
Known Names

Molecular Properties

474.4
MW (Da)
5.87
ALogP
6
HBA
2
HBD
68.3
PSA (Ų)
0.31
QED
1
Ro5 Violations
8
Rot. Bonds

Drug Information

Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C21H20F6N4O2
MW 474.41
Aromatic Rings 3
Heavy Atoms 33
NP-Likeness -1.46

Activity Summary

EC50 1 meas. best 7.0

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Human coronavirus OC43
CHEMBL5209665
EC50 7.0 7.0 100.0 1

Activity Data Samples

Top measurements by pChEMBL value

Literature References

PubMed DOI Target Context # Activities
37813064 10.1016/j.ejmech.2023.115831 Human coronavirus OC43 4
37813064 10.1016/j.ejmech.2023.115831 NCI-H460 1
37813064 10.1016/j.ejmech.2023.115831 ADMET 1

Data from ChEMBL 36 via Core Engine