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Compound Detail

CHEMBL591363

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CC(=O)NC(c1ccc(Cl)cc1)c1ccc2cccnc2c1O

Basic Information

ChEMBL ID CHEMBL591363
Phase Preclinical
Structure Type MOL
InChI Key IXRHAWQJTWGCCU-UHFFFAOYSA-N
2
Targets
2
Activities
1
Assay Types
0
PK Parameters
1
Publications
0
Known Names

Molecular Properties

326.8
MW (Da)
3.82
ALogP
3
HBA
2
HBD
62.2
PSA (Ų)
0.77
QED
0
Ro5 Violations
3
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C18H15ClN2O2
MW 326.78
Aromatic Rings 3
Heavy Atoms 23
NP-Likeness -1.02

Activity Summary

IC50 2 meas. best 4.16

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Unchecked
CHEMBL612545
IC50 4.16 4.16 69866.0 1
No relevant target
CHEMBL2362975
IC50 4.11 4.11 78511.0 1

Activity Data Samples

Top measurements by pChEMBL value

Literature References

PubMed DOI Target Context # Activities
20485428 10.1038/nature09099 Plasmodium falciparum 2

Data from ChEMBL 36 via Core Engine