Assay Detail
Functional
CHEMBL2354263
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PubChem BioAssay. Absorbance-based bacterial cell-based high throughput dose response assay to identify inhibitors of RecBCD. (Class of assay: confirmatory)
130
Total Activities
127
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 130 | 4.29 | 4.83 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1427717 | — | — | 1 | 4.83 |
| CHEMBL1400446 | — | — | 1 | 4.74 |
| CHEMBL187866 | — | — | 1 | 4.73 |
| CHEMBL1474782 | — | — | 1 | 4.73 |
| CHEMBL1969543 | — | — | 1 | 4.68 |
| CHEMBL572994 | — | — | 1 | 4.66 |
| CHEMBL1899240 | — | — | 1 | 4.64 |
| CHEMBL1460853 | — | — | 1 | 4.57 |
| CHEMBL1735962 | — | — | 1 | 4.57 |
| CHEMBL1596605 | — | — | 1 | 4.53 |
| CHEMBL1422429 | — | — | 1 | 4.52 |
| CHEMBL1362047 | — | — | 1 | 4.50 |
| CHEMBL316589 | — | — | 1 | 4.47 |
| CHEMBL1867000 | — | — | 1 | 4.39 |
| CHEMBL1985082 | — | — | 1 | 4.39 |
| CHEMBL1329129 | — | — | 1 | 4.36 |
| CHEMBL1454391 | — | — | 1 | 4.34 |
| CHEMBL1608727 | — | — | 1 | 4.33 |
| CHEMBL1541943 | — | — | 1 | 4.31 |
| CHEMBL1970585 | — | — | 1 | 4.29 |
| CHEMBL991 | STAVUDINE | 4.0 | 3 | 4.28 |
| CHEMBL496 | HEXACHLOROPHENE | 4.0 | 1 | 4.27 |
| CHEMBL1200688 | ERYTHROMYCIN ETHYLSUCCINATE | 4.0 | 1 | 4.27 |
| CHEMBL1443407 | — | — | 1 | 4.24 |
| CHEMBL23970 | — | — | 1 | 4.22 |
| CHEMBL1885868 | — | — | 1 | 4.21 |
| CHEMBL1604735 | — | — | 1 | 4.21 |
| CHEMBL187263 | — | — | 1 | 4.20 |
| CHEMBL1971965 | — | — | 1 | 4.20 |
| CHEMBL1528479 | — | — | 1 | 4.20 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1427717 | — | IC50 | = | 14619.0 | nM | 4.83 |
| CHEMBL1400446 | — | IC50 | = | 18320.0 | nM | 4.74 |
| CHEMBL1474782 | — | IC50 | = | 18557.0 | nM | 4.73 |
| CHEMBL187866 | — | IC50 | = | 18643.0 | nM | 4.73 |
| CHEMBL1969543 | — | IC50 | = | 20684.0 | nM | 4.68 |
| CHEMBL572994 | — | IC50 | = | 21825.0 | nM | 4.66 |
| CHEMBL1899240 | — | IC50 | = | 23101.0 | nM | 4.64 |
| CHEMBL1735962 | — | IC50 | = | 26913.0 | nM | 4.57 |
| CHEMBL1460853 | — | IC50 | = | 26743.0 | nM | 4.57 |
| CHEMBL1596605 | — | IC50 | = | 29742.0 | nM | 4.53 |
| CHEMBL1422429 | — | IC50 | = | 30077.0 | nM | 4.52 |
| CHEMBL1362047 | — | IC50 | = | 31935.0 | nM | 4.50 |
| CHEMBL316589 | — | IC50 | = | 33923.0 | nM | 4.47 |
| CHEMBL1985082 | — | IC50 | = | 40918.0 | nM | 4.39 |
| CHEMBL1867000 | — | IC50 | = | 41156.0 | nM | 4.39 |
| CHEMBL1329129 | — | IC50 | = | 43514.0 | nM | 4.36 |
| CHEMBL1454391 | — | IC50 | = | 45776.0 | nM | 4.34 |
| CHEMBL1608727 | — | IC50 | = | 47123.0 | nM | 4.33 |
| CHEMBL1541943 | — | IC50 | = | 48479.0 | nM | 4.31 |
| CHEMBL1970585 | — | IC50 | = | 51578.0 | nM | 4.29 |
| CHEMBL991 | STAVUDINE | IC50 | = | 52939.0 | nM | 4.28 |
| CHEMBL496 | HEXACHLOROPHENE | IC50 | = | 53344.0 | nM | 4.27 |
| CHEMBL1200688 | ERYTHROMYCIN ETHYLSUCCINATE | IC50 | = | 54233.0 | nM | 4.27 |
| CHEMBL1443407 | — | IC50 | = | 57799.0 | nM | 4.24 |
| CHEMBL991 | STAVUDINE | IC50 | = | 60254.0 | nM | 4.22 |
| CHEMBL23970 | — | IC50 | = | 60506.0 | nM | 4.22 |
| CHEMBL1885868 | — | IC50 | = | 61289.0 | nM | 4.21 |
| CHEMBL1604735 | — | IC50 | = | 61196.0 | nM | 4.21 |
| CHEMBL1971965 | — | IC50 | = | 62468.0 | nM | 4.20 |
| CHEMBL187263 | — | IC50 | = | 63475.0 | nM | 4.20 |
| CHEMBL1528479 | — | IC50 | = | 63537.0 | nM | 4.20 |
| CHEMBL3198603 | — | IC50 | = | 63967.0 | nM | 4.19 |
| CHEMBL1443577 | SULFACHLORPYRIDAZINE | IC50 | = | 64050.0 | nM | 4.19 |
| CHEMBL1129 | TRIFLURIDINE | IC50 | = | 66082.0 | nM | 4.18 |
| CHEMBL1734467 | — | IC50 | = | 66923.0 | nM | 4.17 |
| CHEMBL591363 | — | IC50 | = | 69866.0 | nM | 4.16 |
| CHEMBL991 | STAVUDINE | IC50 | = | 72483.0 | nM | 4.14 |
| CHEMBL2143575 | — | IC50 | = | 72527.0 | nM | 4.14 |
| CHEMBL1905996 | — | IC50 | = | 76239.0 | nM | 4.12 |
| CHEMBL318153 | EDOXUDINE | IC50 | = | 75823.0 | nM | 4.12 |
| CHEMBL437 | SULFATHIAZOLE | IC50 | = | 75908.0 | nM | 4.12 |
| CHEMBL1489217 | — | IC50 | = | 79834.0 | nM | 4.10 |
| CHEMBL2132242 | — | IC50 | = | 85234.0 | nM | 4.07 |
| CHEMBL2135968 | — | IC50 | = | 85688.0 | nM | 4.07 |
| CHEMBL3145315 | — | IC50 | = | 84729.0 | nM | 4.07 |
| CHEMBL1724744 | — | IC50 | = | 87291.0 | nM | 4.06 |
| CHEMBL3197024 | — | IC50 | = | 86239.0 | nM | 4.06 |
| CHEMBL1191 | SULFAMETHIZOLE | IC50 | = | 86564.0 | nM | 4.06 |
| CHEMBL1530766 | — | IC50 | = | 90669.0 | nM | 4.04 |
| CHEMBL443 | SULFAMETHOXAZOLE | IC50 | = | 94317.0 | nM | 4.03 |