Assay Detail
Functional
CHEMBL2354261
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PubChem BioAssay. Counterscreen for inhibitors of RecBCD: Absorbance-based cell-based high throughput dose response assay to identify inhibitors of bacterial viability. (Class of assay: confirmatory)
130
Total Activities
127
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 130 | 4.30 | 4.83 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1427717 | — | — | 1 | 4.83 |
| CHEMBL1474782 | — | — | 1 | 4.74 |
| CHEMBL1400446 | — | — | 1 | 4.73 |
| CHEMBL1969543 | — | — | 1 | 4.70 |
| CHEMBL187866 | — | — | 1 | 4.67 |
| CHEMBL991 | STAVUDINE | 4.0 | 3 | 4.57 |
| CHEMBL1460853 | — | — | 1 | 4.57 |
| CHEMBL316589 | — | — | 1 | 4.54 |
| CHEMBL1362047 | — | — | 1 | 4.51 |
| CHEMBL1899240 | — | — | 1 | 4.49 |
| CHEMBL1443577 | SULFACHLORPYRIDAZINE | 2.0 | 1 | 4.49 |
| CHEMBL1596605 | — | — | 1 | 4.43 |
| CHEMBL1970585 | — | — | 1 | 4.41 |
| CHEMBL572994 | — | — | 1 | 4.39 |
| CHEMBL1867000 | — | — | 1 | 4.38 |
| CHEMBL1604735 | — | — | 1 | 4.36 |
| CHEMBL1443407 | — | — | 1 | 4.36 |
| CHEMBL1422429 | — | — | 1 | 4.35 |
| CHEMBL1735962 | — | — | 1 | 4.35 |
| CHEMBL1329129 | — | — | 1 | 4.34 |
| CHEMBL1454391 | — | — | 1 | 4.33 |
| CHEMBL1608727 | — | — | 1 | 4.29 |
| CHEMBL1541943 | — | — | 1 | 4.29 |
| CHEMBL437 | SULFATHIAZOLE | 4.0 | 1 | 4.28 |
| CHEMBL1985082 | — | — | 1 | 4.27 |
| CHEMBL443 | SULFAMETHOXAZOLE | 4.0 | 1 | 4.27 |
| CHEMBL187263 | — | — | 1 | 4.26 |
| CHEMBL1885868 | — | — | 1 | 4.24 |
| CHEMBL1191 | SULFAMETHIZOLE | 4.0 | 1 | 4.24 |
| CHEMBL1457229 | — | — | 1 | 4.22 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1427717 | — | IC50 | = | 14705.0 | nM | 4.83 |
| CHEMBL1474782 | — | IC50 | = | 18277.0 | nM | 4.74 |
| CHEMBL1400446 | — | IC50 | = | 18796.0 | nM | 4.73 |
| CHEMBL1969543 | — | IC50 | = | 19901.0 | nM | 4.70 |
| CHEMBL187866 | — | IC50 | = | 21622.0 | nM | 4.67 |
| CHEMBL1460853 | — | IC50 | = | 26725.0 | nM | 4.57 |
| CHEMBL991 | STAVUDINE | IC50 | = | 26784.0 | nM | 4.57 |
| CHEMBL316589 | — | IC50 | = | 28627.0 | nM | 4.54 |
| CHEMBL1362047 | — | IC50 | = | 30569.0 | nM | 4.51 |
| CHEMBL1443577 | SULFACHLORPYRIDAZINE | IC50 | = | 32646.0 | nM | 4.49 |
| CHEMBL1899240 | — | IC50 | = | 32307.0 | nM | 4.49 |
| CHEMBL991 | STAVUDINE | IC50 | = | 36024.0 | nM | 4.44 |
| CHEMBL1596605 | — | IC50 | = | 36984.0 | nM | 4.43 |
| CHEMBL1970585 | — | IC50 | = | 38644.0 | nM | 4.41 |
| CHEMBL572994 | — | IC50 | = | 41136.0 | nM | 4.39 |
| CHEMBL1867000 | — | IC50 | = | 41728.0 | nM | 4.38 |
| CHEMBL1443407 | — | IC50 | = | 44086.0 | nM | 4.36 |
| CHEMBL1604735 | — | IC50 | = | 44081.0 | nM | 4.36 |
| CHEMBL1422429 | — | IC50 | = | 44212.0 | nM | 4.35 |
| CHEMBL1735962 | — | IC50 | = | 45019.0 | nM | 4.35 |
| CHEMBL1329129 | — | IC50 | = | 45353.0 | nM | 4.34 |
| CHEMBL1454391 | — | IC50 | = | 46448.0 | nM | 4.33 |
| CHEMBL1541943 | — | IC50 | = | 50990.0 | nM | 4.29 |
| CHEMBL1608727 | — | IC50 | = | 51831.0 | nM | 4.29 |
| CHEMBL437 | SULFATHIAZOLE | IC50 | = | 52095.0 | nM | 4.28 |
| CHEMBL1985082 | — | IC50 | = | 53999.0 | nM | 4.27 |
| CHEMBL443 | SULFAMETHOXAZOLE | IC50 | = | 54149.0 | nM | 4.27 |
| CHEMBL187263 | — | IC50 | = | 54936.0 | nM | 4.26 |
| CHEMBL1191 | SULFAMETHIZOLE | IC50 | = | 57455.0 | nM | 4.24 |
| CHEMBL1885868 | — | IC50 | = | 57591.0 | nM | 4.24 |
| CHEMBL23970 | — | IC50 | = | 59613.0 | nM | 4.22 |
| CHEMBL1457229 | — | IC50 | = | 60820.0 | nM | 4.22 |
| CHEMBL1200688 | ERYTHROMYCIN ETHYLSUCCINATE | IC50 | = | 61714.0 | nM | 4.21 |
| CHEMBL496 | HEXACHLOROPHENE | IC50 | = | 63363.0 | nM | 4.20 |
| CHEMBL1129 | TRIFLURIDINE | IC50 | = | 63075.0 | nM | 4.20 |
| CHEMBL1571122 | — | IC50 | = | 64384.0 | nM | 4.19 |
| CHEMBL2132242 | — | IC50 | = | 66625.0 | nM | 4.18 |
| CHEMBL1971965 | — | IC50 | = | 66241.0 | nM | 4.18 |
| CHEMBL991 | STAVUDINE | IC50 | = | 66857.0 | nM | 4.17 |
| CHEMBL3195656 | — | IC50 | = | 69998.0 | nM | 4.16 |
| CHEMBL1404493 | — | IC50 | = | 72332.0 | nM | 4.14 |
| CHEMBL1582350 | — | IC50 | = | 74719.0 | nM | 4.13 |
| CHEMBL3145315 | — | IC50 | = | 75976.0 | nM | 4.12 |
| CHEMBL591363 | — | IC50 | = | 78511.0 | nM | 4.11 |
| CHEMBL3145306 | — | IC50 | = | 79176.0 | nM | 4.10 |
| CHEMBL3195045 | — | IC50 | = | 79673.0 | nM | 4.10 |
| CHEMBL1528479 | — | IC50 | = | 82240.0 | nM | 4.08 |
| CHEMBL1543433 | — | IC50 | = | 84879.0 | nM | 4.07 |
| CHEMBL1310196 | — | IC50 | = | 84882.0 | nM | 4.07 |
| CHEMBL1725584 | — | IC50 | = | 86672.0 | nM | 4.06 |